Discovery of 3-(N-phenylsulfamoyl)-l-phenylalanine derivatives as novel and orally available LAT1-selective inhibitors

Shuhei Uesugi, Tomoyuki Tsunemi, Hidenobu Murafuji, Kumiko Kadoshima-Yamaoka, Masao Murakawa, Naoyuki Makita, Urara Tomita, Yukiko Doke, Hiroshi Yukiura, Makoto Koyama, Yasuhiro Hayashi, Kyoko Yamashiro, Kazunori Yoshikiyo, Toshiki Tabata, Hiroshi Maruoka

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DOI
10.1007/s00044-026-03541-6
Published
2026-03-31
Container
Medicinal Chemistry Research
Publisher
Springer Science and Business Media LLC
Open access
unknown

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BibTeX

@article{allodium:10.1007/s00044-026-03541-6,
  title = {Discovery of 3-(N-phenylsulfamoyl)-l-phenylalanine derivatives as novel and orally available LAT1-selective inhibitors},
  author = {Shuhei Uesugi and Tomoyuki Tsunemi and Hidenobu Murafuji and Kumiko Kadoshima-Yamaoka and Masao Murakawa and Naoyuki Makita and Urara Tomita and Yukiko Doke and Hiroshi Yukiura and Makoto Koyama and Yasuhiro Hayashi and Kyoko Yamashiro and Kazunori Yoshikiyo and Toshiki Tabata and Hiroshi Maruoka},
  year = {2026},
  journal = {Medicinal Chemistry Research},
  doi = {10.1007/s00044-026-03541-6},
  url = {https://doi.org/10.1007/s00044-026-03541-6}
}

RIS

TY  - JOUR
TI  - Discovery of 3-(N-phenylsulfamoyl)-l-phenylalanine derivatives as novel and orally available LAT1-selective inhibitors
AU  - Shuhei Uesugi
AU  - Tomoyuki Tsunemi
AU  - Hidenobu Murafuji
AU  - Kumiko Kadoshima-Yamaoka
AU  - Masao Murakawa
AU  - Naoyuki Makita
AU  - Urara Tomita
AU  - Yukiko Doke
AU  - Hiroshi Yukiura
AU  - Makoto Koyama
AU  - Yasuhiro Hayashi
AU  - Kyoko Yamashiro
AU  - Kazunori Yoshikiyo
AU  - Toshiki Tabata
AU  - Hiroshi Maruoka
PY  - 2026
JO  - Medicinal Chemistry Research
DO  - 10.1007/s00044-026-03541-6
UR  - https://doi.org/10.1007/s00044-026-03541-6
ER  - 

APA

Uesugi, S., Tsunemi, T., Murafuji, H., Kadoshima-Yamaoka, K., Murakawa, M., Makita, N., Tomita, U., Doke, Y., Yukiura, H., Koyama, M., Hayashi, Y., Yamashiro, K., Yoshikiyo, K., Tabata, T., & Maruoka, H. (2026). Discovery of 3-(N-phenylsulfamoyl)-l-phenylalanine derivatives as novel and orally available LAT1-selective inhibitors. Medicinal Chemistry Research. https://doi.org/10.1007/s00044-026-03541-6

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