Design, synthesis, and structural characterization of covalent tetrahydroquinoline-based inhibitors of coronavirus 3CLpro

Anastasia A. Pronina, Dmitriy N. Shcherbakov, Artem P. Sanchez-Pimentel, Eugeniya V. Nikitina, Fedor I. Zubkov, Yulia V. Meshkova, Mariya K. Marenina, Nikolay V. Maltsev, Svetlana V. Belenkaya, Vadim O. Trufanov, Ekaterina A. Volosnikova, Anna V. Zaykovskay, Sophia S. Borisevich, Edward M. Khamitov, Dmitriy S. Baev, Egor A. Mustaev, Alexey Yu. Fedorov, Sergey G. Arkhipov, Anna V. Vlaskina, Anastasia R. Nemchinova, Valeriya R. Samygina, Oleg V. Pyankov, Olga Yarovaya, Wei Xu, Nariman F. Salakhutdinov, Mikhail V. Khvostov

Open source

DOI
10.1016/j.bioorg.2026.110402
Published
2026-10
Container
Bioorganic Chemistry
Publisher
Elsevier BV
Open access
unknown

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BibTeX

@article{allodium:10.1016/j.bioorg.2026.110402,
  title = {Design, synthesis, and structural characterization of covalent tetrahydroquinoline-based inhibitors of coronavirus 3CLpro},
  author = {Anastasia A. Pronina and Dmitriy N. Shcherbakov and Artem P. Sanchez-Pimentel and Eugeniya V. Nikitina and Fedor I. Zubkov and Yulia V. Meshkova and Mariya K. Marenina and Nikolay V. Maltsev and Svetlana V. Belenkaya and Vadim O. Trufanov and Ekaterina A. Volosnikova and Anna V. Zaykovskay and Sophia S. Borisevich and Edward M. Khamitov and Dmitriy S. Baev and Egor A. Mustaev and Alexey Yu. Fedorov and Sergey G. Arkhipov and Anna V. Vlaskina and Anastasia R. Nemchinova and Valeriya R. Samygina and Oleg V. Pyankov and Olga Yarovaya and Wei Xu and Nariman F. Salakhutdinov and Mikhail V. Khvostov},
  year = {2026},
  journal = {Bioorganic Chemistry},
  doi = {10.1016/j.bioorg.2026.110402},
  url = {https://doi.org/10.1016/j.bioorg.2026.110402}
}

RIS

TY  - JOUR
TI  - Design, synthesis, and structural characterization of covalent tetrahydroquinoline-based inhibitors of coronavirus 3CLpro
AU  - Anastasia A. Pronina
AU  - Dmitriy N. Shcherbakov
AU  - Artem P. Sanchez-Pimentel
AU  - Eugeniya V. Nikitina
AU  - Fedor I. Zubkov
AU  - Yulia V. Meshkova
AU  - Mariya K. Marenina
AU  - Nikolay V. Maltsev
AU  - Svetlana V. Belenkaya
AU  - Vadim O. Trufanov
AU  - Ekaterina A. Volosnikova
AU  - Anna V. Zaykovskay
AU  - Sophia S. Borisevich
AU  - Edward M. Khamitov
AU  - Dmitriy S. Baev
AU  - Egor A. Mustaev
AU  - Alexey Yu. Fedorov
AU  - Sergey G. Arkhipov
AU  - Anna V. Vlaskina
AU  - Anastasia R. Nemchinova
AU  - Valeriya R. Samygina
AU  - Oleg V. Pyankov
AU  - Olga Yarovaya
AU  - Wei Xu
AU  - Nariman F. Salakhutdinov
AU  - Mikhail V. Khvostov
PY  - 2026
JO  - Bioorganic Chemistry
DO  - 10.1016/j.bioorg.2026.110402
UR  - https://doi.org/10.1016/j.bioorg.2026.110402
ER  - 

APA

Pronina, A. A., Shcherbakov, D. N., Sanchez-Pimentel, A. P., Nikitina, E. V., Zubkov, F. I., Meshkova, Y. V., Marenina, M. K., Maltsev, N. V., Belenkaya, S. V., Trufanov, V. O., Volosnikova, E. A., Zaykovskay, A. V., Borisevich, S. S., Khamitov, E. M., Baev, D. S., Mustaev, E. A., Fedorov, A. Y., Arkhipov, S. G., Vlaskina, A. V., Nemchinova, A. R., Samygina, V. R., Pyankov, O. V., Yarovaya, O., Xu, W., Salakhutdinov, N. F., & Khvostov, M. V. (2026). Design, synthesis, and structural characterization of covalent tetrahydroquinoline-based inhibitors of coronavirus 3CLpro. Bioorganic Chemistry. https://doi.org/10.1016/j.bioorg.2026.110402

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