Design, synthesis and biological evaluation of triazolo[1,5-a]pyrimidinone derivatives as potent and orally efficacious WRN helicase inhibitors for MSI cancer therapy.

Xiong Y, Jiang H, Zhang J, Lu J, Yang J, Lin G, Zhang C, Zhang W, Zeng Q, Shi J, Liu M, Jiang Y, Zhao Q, Wang C, He Y, Che C.

Open source

DOI
10.1016/j.bmc.2026.118777
Published
2026-08-13
Container
Bioorg Med Chem
Publisher
Not recorded
Open access
no

Credibility signals

limited evidence Score 43/100 under policy 1.0.0. This is a metadata assessment, not a judgment of the paper's conclusions.

Show all credibility signals

Cite this work

BibTeX

@article{allodium:10.1016/j.bmc.2026.118777,
  title = {Design, synthesis and biological evaluation of triazolo[1,5-a]pyrimidinone derivatives as potent and orally efficacious WRN helicase inhibitors for MSI cancer therapy.},
  author = {Xiong Y and  Jiang H and  Zhang J and  Lu J and  Yang J and  Lin G and  Zhang C and  Zhang W and  Zeng Q and  Shi J and  Liu M and  Jiang Y and  Zhao Q and  Wang C and  He Y and  Che C.},
  year = {2026},
  journal = {Bioorg Med Chem},
  doi = {10.1016/j.bmc.2026.118777},
  url = {https://doi.org/10.1016/j.bmc.2026.118777}
}

RIS

TY  - JOUR
TI  - Design, synthesis and biological evaluation of triazolo[1,5-a]pyrimidinone derivatives as potent and orally efficacious WRN helicase inhibitors for MSI cancer therapy.
AU  - Xiong Y
AU  -  Jiang H
AU  -  Zhang J
AU  -  Lu J
AU  -  Yang J
AU  -  Lin G
AU  -  Zhang C
AU  -  Zhang W
AU  -  Zeng Q
AU  -  Shi J
AU  -  Liu M
AU  -  Jiang Y
AU  -  Zhao Q
AU  -  Wang C
AU  -  He Y
AU  -  Che C.
PY  - 2026
JO  - Bioorg Med Chem
DO  - 10.1016/j.bmc.2026.118777
UR  - https://doi.org/10.1016/j.bmc.2026.118777
ER  - 

APA

Y, X., H, J., J, Z., J, L., J, Y., G, L., C, Z., W, Z., Q, Z., J, S., M, L., Y, J., Q, Z., C, W., Y, H., & C., C. (2026). Design, synthesis and biological evaluation of triazolo[1,5-a]pyrimidinone derivatives as potent and orally efficacious WRN helicase inhibitors for MSI cancer therapy.. Bioorg Med Chem. https://doi.org/10.1016/j.bmc.2026.118777

Source records