Investigation of morpholine isosters for the development of a potent, selective and metabolically stable mTOR kinase inhibitor

Martina De Pascale, Lukas Bissegger, Chiara Tarantelli, Florent Beaufils, Alessandro Prescimone, Hayget Mohamed Seid Hedad, Omar Kayali, Clara Orbegozo, Luka Raguž, Thorsten Schaefer, Paul Hebeisen, Francesco Bertoni, Matthias P. Wymann, Chiara Borsari

Open source

DOI
10.1016/j.ejmech.2022.115038
Published
2023-02
Container
European Journal of Medicinal Chemistry
Publisher
Elsevier BV
Open access
unknown

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BibTeX

@article{allodium:10.1016/j.ejmech.2022.115038,
  title = {Investigation of morpholine isosters for the development of a potent, selective and metabolically stable mTOR kinase inhibitor},
  author = {Martina De Pascale and Lukas Bissegger and Chiara Tarantelli and Florent Beaufils and Alessandro Prescimone and Hayget Mohamed Seid Hedad and Omar Kayali and Clara Orbegozo and Luka Raguž and Thorsten Schaefer and Paul Hebeisen and Francesco Bertoni and Matthias P. Wymann and Chiara Borsari},
  year = {2023},
  journal = {European Journal of Medicinal Chemistry},
  doi = {10.1016/j.ejmech.2022.115038},
  url = {https://doi.org/10.1016/j.ejmech.2022.115038}
}

RIS

TY  - JOUR
TI  - Investigation of morpholine isosters for the development of a potent, selective and metabolically stable mTOR kinase inhibitor
AU  - Martina De Pascale
AU  - Lukas Bissegger
AU  - Chiara Tarantelli
AU  - Florent Beaufils
AU  - Alessandro Prescimone
AU  - Hayget Mohamed Seid Hedad
AU  - Omar Kayali
AU  - Clara Orbegozo
AU  - Luka Raguž
AU  - Thorsten Schaefer
AU  - Paul Hebeisen
AU  - Francesco Bertoni
AU  - Matthias P. Wymann
AU  - Chiara Borsari
PY  - 2023
JO  - European Journal of Medicinal Chemistry
DO  - 10.1016/j.ejmech.2022.115038
UR  - https://doi.org/10.1016/j.ejmech.2022.115038
ER  - 

APA

Pascale, M. D., Bissegger, L., Tarantelli, C., Beaufils, F., Prescimone, A., Hedad, H. M. S., Kayali, O., Orbegozo, C., Raguž, L., Schaefer, T., Hebeisen, P., Bertoni, F., Wymann, M. P., & Borsari, C. (2023). Investigation of morpholine isosters for the development of a potent, selective and metabolically stable mTOR kinase inhibitor. European Journal of Medicinal Chemistry. https://doi.org/10.1016/j.ejmech.2022.115038

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