Discovery of novel dihydropteridone derivatives as orally bioavailable PLK1 inhibitors with reduced hERG inhibitory activity for acute myeloid leukemia treatment.

Hou Y, Li S, Ren L, Zhang L, Zhang N, Miao R, Huang Q, Li Z, Hu C, Xi Z, Tong M, Gong P, Zhao Y, Liu Y, Liu J.

Open source

DOI
10.1016/j.ejmech.2025.117480
Published
2025-03-07
Container
Eur J Med Chem
Publisher
Not recorded
Open access
no

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BibTeX

@article{allodium:10.1016/j.ejmech.2025.117480,
  title = {Discovery of novel dihydropteridone derivatives as orally bioavailable PLK1 inhibitors with reduced hERG inhibitory activity for acute myeloid leukemia treatment.},
  author = {Hou Y and  Li S and  Ren L and  Zhang L and  Zhang N and  Miao R and  Huang Q and  Li Z and  Hu C and  Xi Z and  Tong M and  Gong P and  Zhao Y and  Liu Y and  Liu J.},
  year = {2025},
  journal = {Eur J Med Chem},
  doi = {10.1016/j.ejmech.2025.117480},
  url = {https://doi.org/10.1016/j.ejmech.2025.117480}
}

RIS

TY  - JOUR
TI  - Discovery of novel dihydropteridone derivatives as orally bioavailable PLK1 inhibitors with reduced hERG inhibitory activity for acute myeloid leukemia treatment.
AU  - Hou Y
AU  -  Li S
AU  -  Ren L
AU  -  Zhang L
AU  -  Zhang N
AU  -  Miao R
AU  -  Huang Q
AU  -  Li Z
AU  -  Hu C
AU  -  Xi Z
AU  -  Tong M
AU  -  Gong P
AU  -  Zhao Y
AU  -  Liu Y
AU  -  Liu J.
PY  - 2025
JO  - Eur J Med Chem
DO  - 10.1016/j.ejmech.2025.117480
UR  - https://doi.org/10.1016/j.ejmech.2025.117480
ER  - 

APA

Y, H., S, L., L, R., L, Z., N, Z., R, M., Q, H., Z, L., C, H., Z, X., M, T., P, G., Y, Z., Y, L., & J., L. (2025). Discovery of novel dihydropteridone derivatives as orally bioavailable PLK1 inhibitors with reduced hERG inhibitory activity for acute myeloid leukemia treatment.. Eur J Med Chem. https://doi.org/10.1016/j.ejmech.2025.117480

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