Discovery of an efficacious 2-ethyl-4-phenylthiazole derivative against acute Chagas disease via multiparametric hit-to-lead optimization and in vivo efficacy.

Dit Lapierre TJWJ, Resende DM, de Melo FDSM, Carvalho AMDS, Oliveira DDDS, Michelan-Duarte S, Chelucci RC, Macruz PD, Diniz LA, Ferreira RS, Continentino AL, Moreira GLDS, Xavier ÍLDS, Longo JPF, Calvet CM, Pilau EJ, Ferreira LLG, Andricopulo AD, Neves BJ, Murta SMF, Bastos IMD, Júnior COR.

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DOI
10.1016/j.ejmech.2026.118888
Published
2026-04-28
Container
Eur J Med Chem
Publisher
Not recorded
Open access
no

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BibTeX

@article{allodium:10.1016/j.ejmech.2026.118888,
  title = {Discovery of an efficacious 2-ethyl-4-phenylthiazole derivative against acute Chagas disease via multiparametric hit-to-lead optimization and in vivo efficacy.},
  author = {Dit Lapierre TJWJ and  Resende DM and  de Melo FDSM and  Carvalho AMDS and  Oliveira DDDS and  Michelan-Duarte S and  Chelucci RC and  Macruz PD and  Diniz LA and  Ferreira RS and  Continentino AL and  Moreira GLDS and  Xavier ÍLDS and  Longo JPF and  Calvet CM and  Pilau EJ and  Ferreira LLG and  Andricopulo AD and  Neves BJ and  Murta SMF and  Bastos IMD and  Júnior COR.},
  year = {2026},
  journal = {Eur J Med Chem},
  doi = {10.1016/j.ejmech.2026.118888},
  url = {https://doi.org/10.1016/j.ejmech.2026.118888}
}

RIS

TY  - JOUR
TI  - Discovery of an efficacious 2-ethyl-4-phenylthiazole derivative against acute Chagas disease via multiparametric hit-to-lead optimization and in vivo efficacy.
AU  - Dit Lapierre TJWJ
AU  -  Resende DM
AU  -  de Melo FDSM
AU  -  Carvalho AMDS
AU  -  Oliveira DDDS
AU  -  Michelan-Duarte S
AU  -  Chelucci RC
AU  -  Macruz PD
AU  -  Diniz LA
AU  -  Ferreira RS
AU  -  Continentino AL
AU  -  Moreira GLDS
AU  -  Xavier ÍLDS
AU  -  Longo JPF
AU  -  Calvet CM
AU  -  Pilau EJ
AU  -  Ferreira LLG
AU  -  Andricopulo AD
AU  -  Neves BJ
AU  -  Murta SMF
AU  -  Bastos IMD
AU  -  Júnior COR.
PY  - 2026
JO  - Eur J Med Chem
DO  - 10.1016/j.ejmech.2026.118888
UR  - https://doi.org/10.1016/j.ejmech.2026.118888
ER  - 

APA

TJWJ, D. L., DM, R., FDSM, D. M., AMDS, C., DDDS, O., S, M., RC, C., PD, M., LA, D., RS, F., AL, C., GLDS, M., ÍLDS, X., JPF, L., CM, C., EJ, P., LLG, F., AD, A., BJ, N., SMF, M., IMD, B., & COR., J. (2026). Discovery of an efficacious 2-ethyl-4-phenylthiazole derivative against acute Chagas disease via multiparametric hit-to-lead optimization and in vivo efficacy.. Eur J Med Chem. https://doi.org/10.1016/j.ejmech.2026.118888

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