Leveraging multitargeting BChE-MAO B inhibitors against microglia-related neuroinflammation: in vitro biological evaluation, structure-activity relationships, drug-like properties, and X-ray crystal complexes

Mariagrazia Rullo, Gabriella La Spada, Xavier Brazzolotto, Sara Marchese, Imane Ghafir El Idrissi, Morena Miciaccia, Marco Colella, Jose M. Brea, Eleonora Macchia, Maria I. Loza, Andrea Gottinger, Antonio Scilimati, Maria Grazia Perrone, Angela Stefanachi, Claudia Binda, Francesco Leonetti, Leonardo Pisani

Open source

DOI
10.1016/j.ejmech.2026.118961
Published
2026-10
Container
European Journal of Medicinal Chemistry
Publisher
Elsevier BV
Open access
unknown

Credibility signals

uncertain Score 64/100 under policy 1.0.0. This is a metadata assessment, not a judgment of the paper's conclusions.

Show all credibility signals

Cite this work

BibTeX

@article{allodium:10.1016/j.ejmech.2026.118961,
  title = {Leveraging multitargeting BChE-MAO B inhibitors against microglia-related neuroinflammation: in vitro biological evaluation, structure-activity relationships, drug-like properties, and X-ray crystal complexes},
  author = {Mariagrazia Rullo and Gabriella La Spada and Xavier Brazzolotto and Sara Marchese and Imane Ghafir El Idrissi and Morena Miciaccia and Marco Colella and Jose M. Brea and Eleonora Macchia and Maria I. Loza and Andrea Gottinger and Antonio Scilimati and Maria Grazia Perrone and Angela Stefanachi and Claudia Binda and Francesco Leonetti and Leonardo Pisani},
  year = {2026},
  journal = {European Journal of Medicinal Chemistry},
  doi = {10.1016/j.ejmech.2026.118961},
  url = {https://doi.org/10.1016/j.ejmech.2026.118961}
}

RIS

TY  - JOUR
TI  - Leveraging multitargeting BChE-MAO B inhibitors against microglia-related neuroinflammation: in vitro biological evaluation, structure-activity relationships, drug-like properties, and X-ray crystal complexes
AU  - Mariagrazia Rullo
AU  - Gabriella La Spada
AU  - Xavier Brazzolotto
AU  - Sara Marchese
AU  - Imane Ghafir El Idrissi
AU  - Morena Miciaccia
AU  - Marco Colella
AU  - Jose M. Brea
AU  - Eleonora Macchia
AU  - Maria I. Loza
AU  - Andrea Gottinger
AU  - Antonio Scilimati
AU  - Maria Grazia Perrone
AU  - Angela Stefanachi
AU  - Claudia Binda
AU  - Francesco Leonetti
AU  - Leonardo Pisani
PY  - 2026
JO  - European Journal of Medicinal Chemistry
DO  - 10.1016/j.ejmech.2026.118961
UR  - https://doi.org/10.1016/j.ejmech.2026.118961
ER  - 

APA

Rullo, M., Spada, G. L., Brazzolotto, X., Marchese, S., Idrissi, I. G. E., Miciaccia, M., Colella, M., Brea, J. M., Macchia, E., Loza, M. I., Gottinger, A., Scilimati, A., Perrone, M. G., Stefanachi, A., Binda, C., Leonetti, F., & Pisani, L. (2026). Leveraging multitargeting BChE-MAO B inhibitors against microglia-related neuroinflammation: in vitro biological evaluation, structure-activity relationships, drug-like properties, and X-ray crystal complexes. European Journal of Medicinal Chemistry. https://doi.org/10.1016/j.ejmech.2026.118961

Source records