Discovery of 1,4-diaryl-1,3-dihydro-2H-imidazole-2-thione anticonvulsants integrating AMPA receptor antagonism, Na(v)1.2 channel blockade, redox modulation, and favorable pharmacokinetic properties.

Mahmoud S, El-Moselhy TF, El-Bastawissy EA, Abo El Nasr NME, Elbaset MA, Ibrahim MAA, Khan S, Abalkhail T, Barygin OI, Zhigulin AS, Furman VV, Karelina TV, Huang S, Zamponi GW, Sidhom PA

Open source

DOI
10.1016/j.ejmech.2026.119324
Published
2026 Sep 11
Container
European journal of medicinal chemistry
Publisher
Not recorded
Open access
unknown

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BibTeX

@article{allodium:10.1016/j.ejmech.2026.119324,
  title = {Discovery of 1,4-diaryl-1,3-dihydro-2H-imidazole-2-thione anticonvulsants integrating AMPA receptor antagonism, Na(v)1.2 channel blockade, redox modulation, and favorable pharmacokinetic properties.},
  author = {Mahmoud S and El-Moselhy TF and El-Bastawissy EA and Abo El Nasr NME and Elbaset MA and Ibrahim MAA and Khan S and Abalkhail T and Barygin OI and Zhigulin AS and Furman VV and Karelina TV and Huang S and Zamponi GW and Sidhom PA},
  year = {2026},
  journal = {European journal of medicinal chemistry},
  doi = {10.1016/j.ejmech.2026.119324},
  url = {https://doi.org/10.1016/j.ejmech.2026.119324}
}

RIS

TY  - JOUR
TI  - Discovery of 1,4-diaryl-1,3-dihydro-2H-imidazole-2-thione anticonvulsants integrating AMPA receptor antagonism, Na(v)1.2 channel blockade, redox modulation, and favorable pharmacokinetic properties.
AU  - Mahmoud S
AU  - El-Moselhy TF
AU  - El-Bastawissy EA
AU  - Abo El Nasr NME
AU  - Elbaset MA
AU  - Ibrahim MAA
AU  - Khan S
AU  - Abalkhail T
AU  - Barygin OI
AU  - Zhigulin AS
AU  - Furman VV
AU  - Karelina TV
AU  - Huang S
AU  - Zamponi GW
AU  - Sidhom PA
PY  - 2026
JO  - European journal of medicinal chemistry
DO  - 10.1016/j.ejmech.2026.119324
UR  - https://doi.org/10.1016/j.ejmech.2026.119324
ER  - 

APA

S, M., TF, E., EA, E., NME, A. E. N., MA, E., MAA, I., S, K., T, A., OI, B., AS, Z., VV, F., TV, K., S, H., GW, Z., & PA, S. (2026). Discovery of 1,4-diaryl-1,3-dihydro-2H-imidazole-2-thione anticonvulsants integrating AMPA receptor antagonism, Na(v)1.2 channel blockade, redox modulation, and favorable pharmacokinetic properties.. European journal of medicinal chemistry. https://doi.org/10.1016/j.ejmech.2026.119324

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