Formulation of amorphous solid dispersion of clofazimine, an extremely water-insoluble basic drug, via hot-melt extrusion by applying acid-base supersolubilization principle

Mufaddal H. Kathawala, Hari P. Kandagatla, Alex Avdeef, Martin Kuentz, Tatjana Ž. Verbić, Abu T.M. Serajuddin

Open source

DOI
10.1016/j.ijpharm.2026.127063
Published
2026-07
Container
International Journal of Pharmaceutics
Publisher
Elsevier BV
Open access
unknown

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BibTeX

@article{allodium:10.1016/j.ijpharm.2026.127063,
  title = {Formulation of amorphous solid dispersion of clofazimine, an extremely water-insoluble basic drug, via hot-melt extrusion by applying acid-base supersolubilization principle},
  author = {Mufaddal H. Kathawala and Hari P. Kandagatla and Alex Avdeef and Martin Kuentz and Tatjana Ž. Verbić and Abu T.M. Serajuddin},
  year = {2026},
  journal = {International Journal of Pharmaceutics},
  doi = {10.1016/j.ijpharm.2026.127063},
  url = {https://doi.org/10.1016/j.ijpharm.2026.127063}
}

RIS

TY  - JOUR
TI  - Formulation of amorphous solid dispersion of clofazimine, an extremely water-insoluble basic drug, via hot-melt extrusion by applying acid-base supersolubilization principle
AU  - Mufaddal H. Kathawala
AU  - Hari P. Kandagatla
AU  - Alex Avdeef
AU  - Martin Kuentz
AU  - Tatjana Ž. Verbić
AU  - Abu T.M. Serajuddin
PY  - 2026
JO  - International Journal of Pharmaceutics
DO  - 10.1016/j.ijpharm.2026.127063
UR  - https://doi.org/10.1016/j.ijpharm.2026.127063
ER  - 

APA

Kathawala, M. H., Kandagatla, H. P., Avdeef, A., Kuentz, M., Verbić, T. Ž., & Serajuddin, A. T. (2026). Formulation of amorphous solid dispersion of clofazimine, an extremely water-insoluble basic drug, via hot-melt extrusion by applying acid-base supersolubilization principle. International Journal of Pharmaceutics. https://doi.org/10.1016/j.ijpharm.2026.127063

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