Discovery of tankyrase scaffolding inhibitor specifically targeting the ARC4 peptide binding domain

Chiara Bosetti, Albert Galera-Prat, Sven T. Sowa, Alexandra Gade, Cláudia Braga, Shoshy A. Brinch, Faranak Nami, Johan Pääkkönen, Veeti Pulju, Maureen T. Meling, Maria Candamo-Lourido, Jo Waaler, Mads H. Clausen, Lari Lehtiö

Open source

DOI
10.1016/j.str.2025.12.015
Published
2026-03
Container
Structure
Publisher
Elsevier BV
Open access
unknown

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BibTeX

@article{allodium:10.1016/j.str.2025.12.015,
  title = {Discovery of tankyrase scaffolding inhibitor specifically targeting the ARC4 peptide binding domain},
  author = {Chiara Bosetti and Albert Galera-Prat and Sven T. Sowa and Alexandra Gade and Cláudia Braga and Shoshy A. Brinch and Faranak Nami and Johan Pääkkönen and Veeti Pulju and Maureen T. Meling and Maria Candamo-Lourido and Jo Waaler and Mads H. Clausen and Lari Lehtiö},
  year = {2026},
  journal = {Structure},
  doi = {10.1016/j.str.2025.12.015},
  url = {https://doi.org/10.1016/j.str.2025.12.015}
}

RIS

TY  - JOUR
TI  - Discovery of tankyrase scaffolding inhibitor specifically targeting the ARC4 peptide binding domain
AU  - Chiara Bosetti
AU  - Albert Galera-Prat
AU  - Sven T. Sowa
AU  - Alexandra Gade
AU  - Cláudia Braga
AU  - Shoshy A. Brinch
AU  - Faranak Nami
AU  - Johan Pääkkönen
AU  - Veeti Pulju
AU  - Maureen T. Meling
AU  - Maria Candamo-Lourido
AU  - Jo Waaler
AU  - Mads H. Clausen
AU  - Lari Lehtiö
PY  - 2026
JO  - Structure
DO  - 10.1016/j.str.2025.12.015
UR  - https://doi.org/10.1016/j.str.2025.12.015
ER  - 

APA

Bosetti, C., Galera-Prat, A., Sowa, S. T., Gade, A., Braga, C., Brinch, S. A., Nami, F., Pääkkönen, J., Pulju, V., Meling, M. T., Candamo-Lourido, M., Waaler, J., Clausen, M. H., & Lehtiö, L. (2026). Discovery of tankyrase scaffolding inhibitor specifically targeting the ARC4 peptide binding domain. Structure. https://doi.org/10.1016/j.str.2025.12.015

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