A Chemical Probe for Dark Kinase STK17B Derives Its Potency and High Selectivity through a Unique P-Loop Conformation

Alfredo Picado, Apirat Chaikuad, Carrow I. Wells, Safal Shrestha, William J. Zuercher, Julie E. Pickett, Frank E. Kwarcinski, Parvathi Sinha, Chandi S. de Silva, Reena Zutshi, Shubin Liu, Natarajan Kannan, Stefan Knapp, David H. Drewry, Timothy M. Willson

Open source

DOI
10.1021/acs.jmedchem.0c01174
Published
2020-11-20
Container
Journal of Medicinal Chemistry
Publisher
American Chemical Society (ACS)
Open access
unknown

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BibTeX

@article{allodium:10.1021/acs.jmedchem.0c01174,
  title = {A Chemical Probe for Dark Kinase STK17B Derives Its Potency and High Selectivity through a Unique P-Loop Conformation},
  author = {Alfredo Picado and Apirat Chaikuad and Carrow I. Wells and Safal Shrestha and William J. Zuercher and Julie E. Pickett and Frank E. Kwarcinski and Parvathi Sinha and Chandi S. de Silva and Reena Zutshi and Shubin Liu and Natarajan Kannan and Stefan Knapp and David H. Drewry and Timothy M. Willson},
  year = {2020},
  journal = {Journal of Medicinal Chemistry},
  doi = {10.1021/acs.jmedchem.0c01174},
  url = {https://doi.org/10.1021/acs.jmedchem.0c01174}
}

RIS

TY  - JOUR
TI  - A Chemical Probe for Dark Kinase STK17B Derives Its Potency and High Selectivity through a Unique P-Loop Conformation
AU  - Alfredo Picado
AU  - Apirat Chaikuad
AU  - Carrow I. Wells
AU  - Safal Shrestha
AU  - William J. Zuercher
AU  - Julie E. Pickett
AU  - Frank E. Kwarcinski
AU  - Parvathi Sinha
AU  - Chandi S. de Silva
AU  - Reena Zutshi
AU  - Shubin Liu
AU  - Natarajan Kannan
AU  - Stefan Knapp
AU  - David H. Drewry
AU  - Timothy M. Willson
PY  - 2020
JO  - Journal of Medicinal Chemistry
DO  - 10.1021/acs.jmedchem.0c01174
UR  - https://doi.org/10.1021/acs.jmedchem.0c01174
ER  - 

APA

Picado, A., Chaikuad, A., Wells, C. I., Shrestha, S., Zuercher, W. J., Pickett, J. E., Kwarcinski, F. E., Sinha, P., Silva, C. S. D., Zutshi, R., Liu, S., Kannan, N., Knapp, S., Drewry, D. H., & Willson, T. M. (2020). A Chemical Probe for Dark Kinase STK17B Derives Its Potency and High Selectivity through a Unique P-Loop Conformation. Journal of Medicinal Chemistry. https://doi.org/10.1021/acs.jmedchem.0c01174

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