Structure-Based Discovery of a Series of Covalent, Orally Bioavailable, and Selective BFL1 Inhibitors.

Palisse A, Cheung T, Blokhuis A, Cogswell T, Martins BS, Riemens R, Schellekens R, Battocchio G, Jansen C, Cottee MA, Ornell K, Sacchetto C, Leon L, van Hoek-Emmelot M, Bostock M, Brauer BL, Beaumont K, Lucas SCC, Ahmed S, Blackwell JH, Börjesson U, Gohlke A, Gramatikov IMT, Hargreaves D, van Hoeven V, Kantae V, Kupcova L, Milbradt AG, Seneviratne U, Su N, Vales J, Wang H, White MJ, Kinzel O

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DOI: 10.1021/acs.jmedchem.4c01995
Published: 2024 Dec 26
Container: Journal of medicinal chemistry
Publisher: Not recorded
Open access: unknown

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Cite this work

BibTeX

@article{allodium:10.1021/acs.jmedchem.4c01995,
  title = {Structure-Based Discovery of a Series of Covalent, Orally Bioavailable, and Selective BFL1 Inhibitors.},
  author = {Palisse A and Cheung T and Blokhuis A and Cogswell T and Martins BS and Riemens R and Schellekens R and Battocchio G and Jansen C and Cottee MA and Ornell K and Sacchetto C and Leon L and van Hoek-Emmelot M and Bostock M and Brauer BL and Beaumont K and Lucas SCC and Ahmed S and Blackwell JH and Börjesson U and Gohlke A and Gramatikov IMT and Hargreaves D and van Hoeven V and Kantae V and Kupcova L and Milbradt AG and Seneviratne U and Su N and Vales J and Wang H and White MJ and Kinzel O},
  year = {2024},
  journal = {Journal of medicinal chemistry},
  doi = {10.1021/acs.jmedchem.4c01995},
  url = {https://doi.org/10.1021/acs.jmedchem.4c01995}
}

RIS

TY  - JOUR
TI  - Structure-Based Discovery of a Series of Covalent, Orally Bioavailable, and Selective BFL1 Inhibitors.
AU  - Palisse A
AU  - Cheung T
AU  - Blokhuis A
AU  - Cogswell T
AU  - Martins BS
AU  - Riemens R
AU  - Schellekens R
AU  - Battocchio G
AU  - Jansen C
AU  - Cottee MA
AU  - Ornell K
AU  - Sacchetto C
AU  - Leon L
AU  - van Hoek-Emmelot M
AU  - Bostock M
AU  - Brauer BL
AU  - Beaumont K
AU  - Lucas SCC
AU  - Ahmed S
AU  - Blackwell JH
AU  - Börjesson U
AU  - Gohlke A
AU  - Gramatikov IMT
AU  - Hargreaves D
AU  - van Hoeven V
AU  - Kantae V
AU  - Kupcova L
AU  - Milbradt AG
AU  - Seneviratne U
AU  - Su N
AU  - Vales J
AU  - Wang H
AU  - White MJ
AU  - Kinzel O
PY  - 2024
JO  - Journal of medicinal chemistry
DO  - 10.1021/acs.jmedchem.4c01995
UR  - https://doi.org/10.1021/acs.jmedchem.4c01995
ER  -

APA

A, P., T, C., A, B., T, C., BS, M., R, R., R, S., G, B., C, J., MA, C., K, O., C, S., L, L., M, V. H., M, B., BL, B., K, B., SCC, L., S, A., JH, B., U, B., A, G., IMT, G., D, H., V, V. H., V, K., L, K., AG, M., U, S., N, S., J, V., H, W., MJ, W., & O, K. (2024). Structure-Based Discovery of a Series of Covalent, Orally Bioavailable, and Selective BFL1 Inhibitors.. Journal of medicinal chemistry. https://doi.org/10.1021/acs.jmedchem.4c01995

Source records

pubmed · retrieved 2026-11-10T18:13:25.209Z