Discovery, Optimization, and Preclinical Pharmacology of EP652, a METTL3 Inhibitor with Efficacy in Liquid and Solid Tumor Models.

Dutheuil G, Oukoloff K, Korac J, Lenoir F, El Bousmaqui M, Probst N, Lapin A, Nakhabina G, Sorlet C, Parmentier N, Karila D, Ghavtadze N, Casault P, Claridge S, Sapmaz S, Slater MJ, Fraser GL

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DOI
10.1021/acs.jmedchem.4c02225
Published
2025 Feb 13
Container
Journal of medicinal chemistry
Publisher
Not recorded
Open access
unknown

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BibTeX

@article{allodium:10.1021/acs.jmedchem.4c02225,
  title = {Discovery, Optimization, and Preclinical Pharmacology of EP652, a METTL3 Inhibitor with Efficacy in Liquid and Solid Tumor Models.},
  author = {Dutheuil G and Oukoloff K and Korac J and Lenoir F and El Bousmaqui M and Probst N and Lapin A and Nakhabina G and Sorlet C and Parmentier N and Karila D and Ghavtadze N and Casault P and Claridge S and Sapmaz S and Slater MJ and Fraser GL},
  year = {2025},
  journal = {Journal of medicinal chemistry},
  doi = {10.1021/acs.jmedchem.4c02225},
  url = {https://doi.org/10.1021/acs.jmedchem.4c02225}
}

RIS

TY  - JOUR
TI  - Discovery, Optimization, and Preclinical Pharmacology of EP652, a METTL3 Inhibitor with Efficacy in Liquid and Solid Tumor Models.
AU  - Dutheuil G
AU  - Oukoloff K
AU  - Korac J
AU  - Lenoir F
AU  - El Bousmaqui M
AU  - Probst N
AU  - Lapin A
AU  - Nakhabina G
AU  - Sorlet C
AU  - Parmentier N
AU  - Karila D
AU  - Ghavtadze N
AU  - Casault P
AU  - Claridge S
AU  - Sapmaz S
AU  - Slater MJ
AU  - Fraser GL
PY  - 2025
JO  - Journal of medicinal chemistry
DO  - 10.1021/acs.jmedchem.4c02225
UR  - https://doi.org/10.1021/acs.jmedchem.4c02225
ER  - 

APA

G, D., K, O., J, K., F, L., M, E. B., N, P., A, L., G, N., C, S., N, P., D, K., N, G., P, C., S, C., S, S., MJ, S., & GL, F. (2025). Discovery, Optimization, and Preclinical Pharmacology of EP652, a METTL3 Inhibitor with Efficacy in Liquid and Solid Tumor Models.. Journal of medicinal chemistry. https://doi.org/10.1021/acs.jmedchem.4c02225

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