Discovery of Deuterated 3,4-Dihydro-benzo[e][1,4]diazepine-2,5-dione Derivatives as Potent, Selective and Orally Bioavailable ROCK2 Inhibitors.

Li Y, Zhang L, Xu H, Huang Y, Dai Y, Zhu Q, Chen S, Jiang S, Li L, Yang S

Open source

DOI
10.1021/acs.jmedchem.5c03470
Published
2026 Aug 13
Container
Journal of medicinal chemistry
Publisher
Not recorded
Open access
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BibTeX

@article{allodium:10.1021/acs.jmedchem.5c03470,
  title = {Discovery of Deuterated 3,4-Dihydro-benzo[e][1,4]diazepine-2,5-dione Derivatives as Potent, Selective and Orally Bioavailable ROCK2 Inhibitors.},
  author = {Li Y and Zhang L and Xu H and Huang Y and Dai Y and Zhu Q and Chen S and Jiang S and Li L and Yang S},
  year = {2026},
  journal = {Journal of medicinal chemistry},
  doi = {10.1021/acs.jmedchem.5c03470},
  url = {https://doi.org/10.1021/acs.jmedchem.5c03470}
}

RIS

TY  - JOUR
TI  - Discovery of Deuterated 3,4-Dihydro-benzo[e][1,4]diazepine-2,5-dione Derivatives as Potent, Selective and Orally Bioavailable ROCK2 Inhibitors.
AU  - Li Y
AU  - Zhang L
AU  - Xu H
AU  - Huang Y
AU  - Dai Y
AU  - Zhu Q
AU  - Chen S
AU  - Jiang S
AU  - Li L
AU  - Yang S
PY  - 2026
JO  - Journal of medicinal chemistry
DO  - 10.1021/acs.jmedchem.5c03470
UR  - https://doi.org/10.1021/acs.jmedchem.5c03470
ER  - 

APA

Y, L., L, Z., H, X., Y, H., Y, D., Q, Z., S, C., S, J., L, L., & S, Y. (2026). Discovery of Deuterated 3,4-Dihydro-benzo[e][1,4]diazepine-2,5-dione Derivatives as Potent, Selective and Orally Bioavailable ROCK2 Inhibitors.. Journal of medicinal chemistry. https://doi.org/10.1021/acs.jmedchem.5c03470

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