Rapid Identification of a Potent, Selective, and Orally Active p300/CBP Bromodomain Inhibitor Bearing an Imidazo[1,2- <i>a</i> ]pyridine Scaffold via a Highly Efficient Four-Step Synthesis

Zonglong Chen, Ying Zhang, Zihan Li, Hui Shen, Hanqi Wang, Hong Yang, Cheng Zhang, Jiankang Hu, Yujie Wang, Qiongyu Shi, Yan Zhang, Jian Ding, Yanfen Fang, Yong Xu, Xun Huang, Yingxia Li

Open source

DOI
10.1021/acs.jmedchem.5c03730
Published
2026-07-17
Container
Journal of Medicinal Chemistry
Publisher
American Chemical Society (ACS)
Open access
unknown

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BibTeX

@article{allodium:10.1021/acs.jmedchem.5c03730,
  title = {Rapid Identification
of a Potent, Selective, and Orally
Active p300/CBP Bromodomain Inhibitor Bearing an Imidazo[1,2-
                    <i>a</i>
                    ]pyridine Scaffold via a Highly Efficient Four-Step Synthesis},
  author = {Zonglong Chen and Ying Zhang and Zihan Li and Hui Shen and Hanqi Wang and Hong Yang and Cheng Zhang and Jiankang Hu and Yujie Wang and Qiongyu Shi and Yan Zhang and Jian Ding and Yanfen Fang and Yong Xu and Xun Huang and Yingxia Li},
  year = {2026},
  journal = {Journal of Medicinal Chemistry},
  doi = {10.1021/acs.jmedchem.5c03730},
  url = {https://doi.org/10.1021/acs.jmedchem.5c03730}
}

RIS

TY  - JOUR
TI  - Rapid Identification
of a Potent, Selective, and Orally
Active p300/CBP Bromodomain Inhibitor Bearing an Imidazo[1,2-
                    <i>a</i>
                    ]pyridine Scaffold via a Highly Efficient Four-Step Synthesis
AU  - Zonglong Chen
AU  - Ying Zhang
AU  - Zihan Li
AU  - Hui Shen
AU  - Hanqi Wang
AU  - Hong Yang
AU  - Cheng Zhang
AU  - Jiankang Hu
AU  - Yujie Wang
AU  - Qiongyu Shi
AU  - Yan Zhang
AU  - Jian Ding
AU  - Yanfen Fang
AU  - Yong Xu
AU  - Xun Huang
AU  - Yingxia Li
PY  - 2026
JO  - Journal of Medicinal Chemistry
DO  - 10.1021/acs.jmedchem.5c03730
UR  - https://doi.org/10.1021/acs.jmedchem.5c03730
ER  - 

APA

Chen, Z., Zhang, Y., Li, Z., Shen, H., Wang, H., Yang, H., Zhang, C., Hu, J., Wang, Y., Shi, Q., Zhang, Y., Ding, J., Fang, Y., Xu, Y., Huang, X., & Li, Y. (2026). Rapid Identification of a Potent, Selective, and Orally Active p300/CBP Bromodomain Inhibitor Bearing an Imidazo[1,2- <i>a</i> ]pyridine Scaffold via a Highly Efficient Four-Step Synthesis. Journal of Medicinal Chemistry. https://doi.org/10.1021/acs.jmedchem.5c03730

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