Discovery of an Androgen Receptor Degrader Featuring a Pyridazinyl Glutarimide CRBN-Binding Motif for Transdermal Treatment of Androgenetic Alopecia.

Wang X, Ge L, Yu Y, Zhong T, Hu W, Zhang S, Chen X, Yang M, Zhang X, Li Z, Zhuang Z, Zhang S, Jiang X, Wang T, Chen H, Fang S, Gao J, Qin C.

Open source

DOI
10.1021/acs.jmedchem.5c03843
Published
2026-05-29
Container
J Med Chem
Publisher
Not recorded
Open access
no

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BibTeX

@article{allodium:10.1021/acs.jmedchem.5c03843,
  title = {Discovery of an Androgen Receptor Degrader Featuring a Pyridazinyl Glutarimide CRBN-Binding Motif for Transdermal Treatment of Androgenetic Alopecia.},
  author = {Wang X and  Ge L and  Yu Y and  Zhong T and  Hu W and  Zhang S and  Chen X and  Yang M and  Zhang X and  Li Z and  Zhuang Z and  Zhang S and  Jiang X and  Wang T and  Chen H and  Fang S and  Gao J and  Qin C.},
  year = {2026},
  journal = {J Med Chem},
  doi = {10.1021/acs.jmedchem.5c03843},
  url = {https://doi.org/10.1021/acs.jmedchem.5c03843}
}

RIS

TY  - JOUR
TI  - Discovery of an Androgen Receptor Degrader Featuring a Pyridazinyl Glutarimide CRBN-Binding Motif for Transdermal Treatment of Androgenetic Alopecia.
AU  - Wang X
AU  -  Ge L
AU  -  Yu Y
AU  -  Zhong T
AU  -  Hu W
AU  -  Zhang S
AU  -  Chen X
AU  -  Yang M
AU  -  Zhang X
AU  -  Li Z
AU  -  Zhuang Z
AU  -  Zhang S
AU  -  Jiang X
AU  -  Wang T
AU  -  Chen H
AU  -  Fang S
AU  -  Gao J
AU  -  Qin C.
PY  - 2026
JO  - J Med Chem
DO  - 10.1021/acs.jmedchem.5c03843
UR  - https://doi.org/10.1021/acs.jmedchem.5c03843
ER  - 

APA

X, W., L, G., Y, Y., T, Z., W, H., S, Z., X, C., M, Y., X, Z., Z, L., Z, Z., S, Z., X, J., T, W., H, C., S, F., J, G., & C., Q. (2026). Discovery of an Androgen Receptor Degrader Featuring a Pyridazinyl Glutarimide CRBN-Binding Motif for Transdermal Treatment of Androgenetic Alopecia.. J Med Chem. https://doi.org/10.1021/acs.jmedchem.5c03843

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