A Novel Dual-Targeting PROTAC Overcomes Endocrine Resistance by Engaging Orthosteric and Allosteric Sites of Estrogen Receptor α.

Wang C, Xu B, Xin L, Guo Z, Deng X, Dong C, Yang J, Zhou HB.

DOI: 10.1021/acs.jmedchem.6c00521
Published: 2026-08-01
Container: J Med Chem
Publisher: Not recorded
Open access: no

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Cite this work

BibTeX

@article{allodium:10.1021/acs.jmedchem.6c00521,
  title = {A Novel Dual-Targeting PROTAC Overcomes Endocrine Resistance by Engaging Orthosteric and Allosteric Sites of Estrogen Receptor α.},
  author = {Wang C and  Xu B and  Xin L and  Guo Z and  Deng X and  Dong C and  Yang J and  Zhou HB.},
  year = {2026},
  journal = {J Med Chem},
  doi = {10.1021/acs.jmedchem.6c00521},
  url = {https://doi.org/10.1021/acs.jmedchem.6c00521}
}

RIS

TY  - JOUR
TI  - A Novel Dual-Targeting PROTAC Overcomes Endocrine Resistance by Engaging Orthosteric and Allosteric Sites of Estrogen Receptor α.
AU  - Wang C
AU  -  Xu B
AU  -  Xin L
AU  -  Guo Z
AU  -  Deng X
AU  -  Dong C
AU  -  Yang J
AU  -  Zhou HB.
PY  - 2026
JO  - J Med Chem
DO  - 10.1021/acs.jmedchem.6c00521
UR  - https://doi.org/10.1021/acs.jmedchem.6c00521
ER  -

APA

C, W., B, X., L, X., Z, G., X, D., C, D., J, Y., & HB., Z. (2026). A Novel Dual-Targeting PROTAC Overcomes Endocrine Resistance by Engaging Orthosteric and Allosteric Sites of Estrogen Receptor α.. J Med Chem. https://doi.org/10.1021/acs.jmedchem.6c00521

Source records

europe-pmc · retrieved 2026-09-27T14:36:14.977Z