Integrating AI in Medicinal Chemistry for Accelerated Drug Discovery: A Comprehensive SAR (CSAR) Optimization Strategy and Discovery of Potent ALDH3A1 Inhibitors.

Jain S, Yasgar A, Dalal A, Nilova A, Davies M, Baljinnyam B, Qu Y, Denson JP, Esposito D, Tao D, Yang SM, Talley DC, Simeonov A, Martinez NJ, Rai G, Zakharov AV

Open source

DOI
10.1021/acs.jmedchem.6c00537
Published
2026 Jun 11
Container
Journal of medicinal chemistry
Publisher
Not recorded
Open access
yes

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BibTeX

@article{allodium:10.1021/acs.jmedchem.6c00537,
  title = {Integrating AI in Medicinal Chemistry for Accelerated Drug Discovery: A Comprehensive SAR (CSAR) Optimization Strategy and Discovery of Potent ALDH3A1 Inhibitors.},
  author = {Jain S and Yasgar A and Dalal A and Nilova A and Davies M and Baljinnyam B and Qu Y and Denson JP and Esposito D and Tao D and Yang SM and Talley DC and Simeonov A and Martinez NJ and Rai G and Zakharov AV},
  year = {2026},
  journal = {Journal of medicinal chemistry},
  doi = {10.1021/acs.jmedchem.6c00537},
  url = {https://doi.org/10.1021/acs.jmedchem.6c00537}
}

RIS

TY  - JOUR
TI  - Integrating AI in Medicinal Chemistry for Accelerated Drug Discovery: A Comprehensive SAR (CSAR) Optimization Strategy and Discovery of Potent ALDH3A1 Inhibitors.
AU  - Jain S
AU  - Yasgar A
AU  - Dalal A
AU  - Nilova A
AU  - Davies M
AU  - Baljinnyam B
AU  - Qu Y
AU  - Denson JP
AU  - Esposito D
AU  - Tao D
AU  - Yang SM
AU  - Talley DC
AU  - Simeonov A
AU  - Martinez NJ
AU  - Rai G
AU  - Zakharov AV
PY  - 2026
JO  - Journal of medicinal chemistry
DO  - 10.1021/acs.jmedchem.6c00537
UR  - https://doi.org/10.1021/acs.jmedchem.6c00537
ER  - 

APA

S, J., A, Y., A, D., A, N., M, D., B, B., Y, Q., JP, D., D, E., D, T., SM, Y., DC, T., A, S., NJ, M., G, R., & AV, Z. (2026). Integrating AI in Medicinal Chemistry for Accelerated Drug Discovery: A Comprehensive SAR (CSAR) Optimization Strategy and Discovery of Potent ALDH3A1 Inhibitors.. Journal of medicinal chemistry. https://doi.org/10.1021/acs.jmedchem.6c00537

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