Discovery of Highly Potent and Selective, Orally Bioavailable BTK-Targeting PROTACs Featuring Novel CRBN-Binding Warheads.
- DOI
- 10.1021/acs.jmedchem.6c01136
- Published
- 2026 Sep 10
- Container
- Journal of medicinal chemistry
- Publisher
- Not recorded
- Open access
- unknown
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Cite this work
BibTeX
@article{allodium:10.1021/acs.jmedchem.6c01136,
title = {Discovery of Highly Potent and Selective, Orally Bioavailable BTK-Targeting PROTACs Featuring Novel CRBN-Binding Warheads.},
author = {Mantsyzov AB and Zhao P and Kruse CG and Petrov R and Huang F and Yu J and Cai X and Ding X and Aladinskiy V and Aliper A and Ren F and Zhavoronkov A},
year = {2026},
journal = {Journal of medicinal chemistry},
doi = {10.1021/acs.jmedchem.6c01136},
url = {https://doi.org/10.1021/acs.jmedchem.6c01136}
}RIS
TY - JOUR TI - Discovery of Highly Potent and Selective, Orally Bioavailable BTK-Targeting PROTACs Featuring Novel CRBN-Binding Warheads. AU - Mantsyzov AB AU - Zhao P AU - Kruse CG AU - Petrov R AU - Huang F AU - Yu J AU - Cai X AU - Ding X AU - Aladinskiy V AU - Aliper A AU - Ren F AU - Zhavoronkov A PY - 2026 JO - Journal of medicinal chemistry DO - 10.1021/acs.jmedchem.6c01136 UR - https://doi.org/10.1021/acs.jmedchem.6c01136 ER -
APA
AB, M., P, Z., CG, K., R, P., F, H., J, Y., X, C., X, D., V, A., A, A., F, R., & A, Z. (2026). Discovery of Highly Potent and Selective, Orally Bioavailable BTK-Targeting PROTACs Featuring Novel CRBN-Binding Warheads.. Journal of medicinal chemistry. https://doi.org/10.1021/acs.jmedchem.6c01136
Source records
- pubmed · retrieved 2026-09-25T23:13:00.861Z