Discovery of GPCR Antagonists with Potent In Vitro and In Vivo Macrofilaricidal Activity.

Rosa BA, Han Z, Arun A, Tricoche N, Peguero R, Banas V, Shadrick M, Fath M, Suksomboon P, Bharti S, Bancks M, Rehborg EG, Zamanian M, Cho-Ngwa F, Lustigman S, Janetka JW, Mitreva M

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DOI: 10.1021/acs.jmedchem.6c01435
Published: 2026 Aug 13
Container: Journal of medicinal chemistry
Publisher: Not recorded
Open access: unknown

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Cite this work

BibTeX

@article{allodium:10.1021/acs.jmedchem.6c01435,
  title = {Discovery of GPCR Antagonists with Potent In Vitro and In Vivo Macrofilaricidal Activity.},
  author = {Rosa BA and Han Z and Arun A and Tricoche N and Peguero R and Banas V and Shadrick M and Fath M and Suksomboon P and Bharti S and Bancks M and Rehborg EG and Zamanian M and Cho-Ngwa F and Lustigman S and Janetka JW and Mitreva M},
  year = {2026},
  journal = {Journal of medicinal chemistry},
  doi = {10.1021/acs.jmedchem.6c01435},
  url = {https://doi.org/10.1021/acs.jmedchem.6c01435}
}

RIS

TY  - JOUR
TI  - Discovery of GPCR Antagonists with Potent In Vitro and In Vivo Macrofilaricidal Activity.
AU  - Rosa BA
AU  - Han Z
AU  - Arun A
AU  - Tricoche N
AU  - Peguero R
AU  - Banas V
AU  - Shadrick M
AU  - Fath M
AU  - Suksomboon P
AU  - Bharti S
AU  - Bancks M
AU  - Rehborg EG
AU  - Zamanian M
AU  - Cho-Ngwa F
AU  - Lustigman S
AU  - Janetka JW
AU  - Mitreva M
PY  - 2026
JO  - Journal of medicinal chemistry
DO  - 10.1021/acs.jmedchem.6c01435
UR  - https://doi.org/10.1021/acs.jmedchem.6c01435
ER  -

APA

BA, R., Z, H., A, A., N, T., R, P., V, B., M, S., M, F., P, S., S, B., M, B., EG, R., M, Z., F, C., S, L., JW, J., & M, M. (2026). Discovery of GPCR Antagonists with Potent In Vitro and In Vivo Macrofilaricidal Activity.. Journal of medicinal chemistry. https://doi.org/10.1021/acs.jmedchem.6c01435

Source records

pubmed · retrieved 2026-09-26T02:47:44.723Z