Trifluoromethylthio and Trifluoromethyl Functionalization of Endomorphin-1 Enhances its Hydrophobicity and Plasma Stability while Preserving its Affinity for the μ-Opioid Receptor.

Gregorc J, De Neve J, Guitot K, Holleran BJ, Lensen N, Gendron L, Brigaud T, Iskra J, Ballet S, Chaume G

Open source

DOI
10.1021/acs.joc.6c00321
Published
2026 Apr 24
Container
The Journal of organic chemistry
Publisher
Not recorded
Open access
yes

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BibTeX

@article{allodium:10.1021/acs.joc.6c00321,
  title = {Trifluoromethylthio and Trifluoromethyl Functionalization of Endomorphin-1 Enhances its Hydrophobicity and Plasma Stability while Preserving its Affinity for the μ-Opioid Receptor.},
  author = {Gregorc J and De Neve J and Guitot K and Holleran BJ and Lensen N and Gendron L and Brigaud T and Iskra J and Ballet S and Chaume G},
  year = {2026},
  journal = {The Journal of organic chemistry},
  doi = {10.1021/acs.joc.6c00321},
  url = {https://doi.org/10.1021/acs.joc.6c00321}
}

RIS

TY  - JOUR
TI  - Trifluoromethylthio and Trifluoromethyl Functionalization of Endomorphin-1 Enhances its Hydrophobicity and Plasma Stability while Preserving its Affinity for the μ-Opioid Receptor.
AU  - Gregorc J
AU  - De Neve J
AU  - Guitot K
AU  - Holleran BJ
AU  - Lensen N
AU  - Gendron L
AU  - Brigaud T
AU  - Iskra J
AU  - Ballet S
AU  - Chaume G
PY  - 2026
JO  - The Journal of organic chemistry
DO  - 10.1021/acs.joc.6c00321
UR  - https://doi.org/10.1021/acs.joc.6c00321
ER  - 

APA

J, G., J, D. N., K, G., BJ, H., N, L., L, G., T, B., J, I., S, B., & G, C. (2026). Trifluoromethylthio and Trifluoromethyl Functionalization of Endomorphin-1 Enhances its Hydrophobicity and Plasma Stability while Preserving its Affinity for the μ-Opioid Receptor.. The Journal of organic chemistry. https://doi.org/10.1021/acs.joc.6c00321

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