Optimization of Indole- and Pyrazole-fused Glycyrrhetinic Acid Derivatives as Potent PTP1B Inhibitors: In Silico, In Vitro, In Vivo, and Metabolomic Studies.

López-Sánchez M, Mendoza-Mota H, De-la-Cruz-Martínez L, Matadamas-Martínez F, Torres-Chacón DL, Martínez-Arellano R, Palacios-Espinosa JF, Pérez-Villanueva J, González-Andrade M, Páez-Franco JC, Almanza-Pérez JC, Cortés-Benítez F

Open source

DOI
10.1021/acsbiomedchemau.5c00164
Published
2026 Feb 18
Container
ACS bio & med chem Au
Publisher
Not recorded
Open access
yes

Credibility signals

limited evidence Score 45/100 under policy 1.0.0. This is a metadata assessment, not a judgment of the paper's conclusions.

Show all credibility signals

Cite this work

BibTeX

@article{allodium:10.1021/acsbiomedchemau.5c00164,
  title = {Optimization of Indole- and Pyrazole-fused Glycyrrhetinic Acid Derivatives as Potent PTP1B Inhibitors: In Silico, In Vitro, In Vivo, and Metabolomic Studies.},
  author = {López-Sánchez M and Mendoza-Mota H and De-la-Cruz-Martínez L and Matadamas-Martínez F and Torres-Chacón DL and Martínez-Arellano R and Palacios-Espinosa JF and Pérez-Villanueva J and González-Andrade M and Páez-Franco JC and Almanza-Pérez JC and Cortés-Benítez F},
  year = {2026},
  journal = {ACS bio \& med chem Au},
  doi = {10.1021/acsbiomedchemau.5c00164},
  url = {https://doi.org/10.1021/acsbiomedchemau.5c00164}
}

RIS

TY  - JOUR
TI  - Optimization of Indole- and Pyrazole-fused Glycyrrhetinic Acid Derivatives as Potent PTP1B Inhibitors: In Silico, In Vitro, In Vivo, and Metabolomic Studies.
AU  - López-Sánchez M
AU  - Mendoza-Mota H
AU  - De-la-Cruz-Martínez L
AU  - Matadamas-Martínez F
AU  - Torres-Chacón DL
AU  - Martínez-Arellano R
AU  - Palacios-Espinosa JF
AU  - Pérez-Villanueva J
AU  - González-Andrade M
AU  - Páez-Franco JC
AU  - Almanza-Pérez JC
AU  - Cortés-Benítez F
PY  - 2026
JO  - ACS bio & med chem Au
DO  - 10.1021/acsbiomedchemau.5c00164
UR  - https://doi.org/10.1021/acsbiomedchemau.5c00164
ER  - 

APA

M, L., H, M., L, D., F, M., DL, T., R, M., JF, P., J, P., M, G., JC, P., JC, A., & F, C. (2026). Optimization of Indole- and Pyrazole-fused Glycyrrhetinic Acid Derivatives as Potent PTP1B Inhibitors: In Silico, In Vitro, In Vivo, and Metabolomic Studies.. ACS bio & med chem Au. https://doi.org/10.1021/acsbiomedchemau.5c00164

Source records