Discovery and Characterization of a Novel Series of Chloropyrimidines as Covalent Inhibitors of the Kinase MSK1

Adrian Hall, Jan Abendroth, Madison J. Bolejack, Tom Ceska, Sylvie Dell’Aiera, Victoria Ellis, David Fox, Cyril François, Muigai M. Muruthi, Camille Prével, Karine Poullennec, Sergei Romanov, Anne Valade, Alain Vanbellinghen, Jason Yano, Martine Geraerts

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DOI
10.1021/acsmedchemlett.2c00134
Published
2022-06-25
Container
ACS Medicinal Chemistry Letters
Publisher
American Chemical Society (ACS)
Open access
unknown

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BibTeX

@article{allodium:10.1021/acsmedchemlett.2c00134,
  title = {Discovery and Characterization of a Novel Series of Chloropyrimidines as Covalent Inhibitors of the Kinase MSK1},
  author = {Adrian Hall and Jan Abendroth and Madison J. Bolejack and Tom Ceska and Sylvie Dell’Aiera and Victoria Ellis and David Fox and Cyril François and Muigai M. Muruthi and Camille Prével and Karine Poullennec and Sergei Romanov and Anne Valade and Alain Vanbellinghen and Jason Yano and Martine Geraerts},
  year = {2022},
  journal = {ACS Medicinal Chemistry Letters},
  doi = {10.1021/acsmedchemlett.2c00134},
  url = {https://doi.org/10.1021/acsmedchemlett.2c00134}
}

RIS

TY  - JOUR
TI  - Discovery and Characterization of a Novel Series of Chloropyrimidines as Covalent Inhibitors of the Kinase MSK1
AU  - Adrian Hall
AU  - Jan Abendroth
AU  - Madison J. Bolejack
AU  - Tom Ceska
AU  - Sylvie Dell’Aiera
AU  - Victoria Ellis
AU  - David Fox
AU  - Cyril François
AU  - Muigai M. Muruthi
AU  - Camille Prével
AU  - Karine Poullennec
AU  - Sergei Romanov
AU  - Anne Valade
AU  - Alain Vanbellinghen
AU  - Jason Yano
AU  - Martine Geraerts
PY  - 2022
JO  - ACS Medicinal Chemistry Letters
DO  - 10.1021/acsmedchemlett.2c00134
UR  - https://doi.org/10.1021/acsmedchemlett.2c00134
ER  - 

APA

Hall, A., Abendroth, J., Bolejack, M. J., Ceska, T., Dell’Aiera, S., Ellis, V., Fox, D., François, C., Muruthi, M. M., Prével, C., Poullennec, K., Romanov, S., Valade, A., Vanbellinghen, A., Yano, J., & Geraerts, M. (2022). Discovery and Characterization of a Novel Series of Chloropyrimidines as Covalent Inhibitors of the Kinase MSK1. ACS Medicinal Chemistry Letters. https://doi.org/10.1021/acsmedchemlett.2c00134

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