Discovery of Potent, Selective, and Brain-Penetrant Small Molecule CD38 Inhibitors

Andrew J. Stott, Roland W. Bürli, Kevin J. Doyle, Louise Dickson, Richard C. Hewer, Philip Pickford, Maxine J. Roberts, Rosie Waters-Hall, Yiming Wu, Matthias Zebisch, Victor Rangel, Matthis Geitmann, Kim Matthews, Nicola L. Brice, Mark Carlton, Lee A. Dawson, Jenna R. M. Harvey

Open source

DOI
10.1021/acsmedchemlett.5c00727
Published
2026-01-29
Container
ACS Medicinal Chemistry Letters
Publisher
American Chemical Society (ACS)
Open access
unknown

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BibTeX

@article{allodium:10.1021/acsmedchemlett.5c00727,
  title = {Discovery of Potent, Selective, and Brain-Penetrant Small Molecule CD38 Inhibitors},
  author = {Andrew J. Stott and Roland W. Bürli and Kevin J. Doyle and Louise Dickson and Richard C. Hewer and Philip Pickford and Maxine J. Roberts and Rosie Waters-Hall and Yiming Wu and Matthias Zebisch and Victor Rangel and Matthis Geitmann and Kim Matthews and Nicola L. Brice and Mark Carlton and Lee A. Dawson and Jenna R. M. Harvey},
  year = {2026},
  journal = {ACS Medicinal Chemistry Letters},
  doi = {10.1021/acsmedchemlett.5c00727},
  url = {https://doi.org/10.1021/acsmedchemlett.5c00727}
}

RIS

TY  - JOUR
TI  - Discovery of Potent, Selective, and Brain-Penetrant Small Molecule CD38 Inhibitors
AU  - Andrew J. Stott
AU  - Roland W. Bürli
AU  - Kevin J. Doyle
AU  - Louise Dickson
AU  - Richard C. Hewer
AU  - Philip Pickford
AU  - Maxine J. Roberts
AU  - Rosie Waters-Hall
AU  - Yiming Wu
AU  - Matthias Zebisch
AU  - Victor Rangel
AU  - Matthis Geitmann
AU  - Kim Matthews
AU  - Nicola L. Brice
AU  - Mark Carlton
AU  - Lee A. Dawson
AU  - Jenna R. M. Harvey
PY  - 2026
JO  - ACS Medicinal Chemistry Letters
DO  - 10.1021/acsmedchemlett.5c00727
UR  - https://doi.org/10.1021/acsmedchemlett.5c00727
ER  - 

APA

Stott, A. J., Bürli, R. W., Doyle, K. J., Dickson, L., Hewer, R. C., Pickford, P., Roberts, M. J., Waters-Hall, R., Wu, Y., Zebisch, M., Rangel, V., Geitmann, M., Matthews, K., Brice, N. L., Carlton, M., Dawson, L. A., & Harvey, J. R. M. (2026). Discovery of Potent, Selective, and Brain-Penetrant Small Molecule CD38 Inhibitors. ACS Medicinal Chemistry Letters. https://doi.org/10.1021/acsmedchemlett.5c00727

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