Discovery of Forvisirvat (DS-7830a/SP-624), a Brain-Penetrant Sirtuin 6 Activator Derived from Griseofulvin with Antidepressant-Like Effects

Yasuyuki Ogawa, Keiji Saito, Katsuyoshi Nakajima, Osamu Iwamoto, Kazumasa Aoki, Mitsuhiro Makino, Shinji Tanaka, Nobuya Kurikawa, Eriko Michishita-Kioi, Seiko Nagata, Yoko Fujita, Masato Sasaki, Akiko Kasahara, Isao Yasumatsu, Makoto Hirasawa, Wataru Saitoh

Open source

DOI
10.1021/acsmedchemlett.6c00366
Published
2026-08-26
Container
ACS Medicinal Chemistry Letters
Publisher
American Chemical Society (ACS)
Open access
unknown

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BibTeX

@article{allodium:10.1021/acsmedchemlett.6c00366,
  title = {Discovery
of Forvisirvat (DS-7830a/SP-624), a Brain-Penetrant
Sirtuin 6 Activator Derived from Griseofulvin with Antidepressant-Like
Effects},
  author = {Yasuyuki Ogawa and Keiji Saito and Katsuyoshi Nakajima and Osamu Iwamoto and Kazumasa Aoki and Mitsuhiro Makino and Shinji Tanaka and Nobuya Kurikawa and Eriko Michishita-Kioi and Seiko Nagata and Yoko Fujita and Masato Sasaki and Akiko Kasahara and Isao Yasumatsu and Makoto Hirasawa and Wataru Saitoh},
  year = {2026},
  journal = {ACS Medicinal Chemistry
Letters},
  doi = {10.1021/acsmedchemlett.6c00366},
  url = {https://doi.org/10.1021/acsmedchemlett.6c00366}
}

RIS

TY  - JOUR
TI  - Discovery
of Forvisirvat (DS-7830a/SP-624), a Brain-Penetrant
Sirtuin 6 Activator Derived from Griseofulvin with Antidepressant-Like
Effects
AU  - Yasuyuki Ogawa
AU  - Keiji Saito
AU  - Katsuyoshi Nakajima
AU  - Osamu Iwamoto
AU  - Kazumasa Aoki
AU  - Mitsuhiro Makino
AU  - Shinji Tanaka
AU  - Nobuya Kurikawa
AU  - Eriko Michishita-Kioi
AU  - Seiko Nagata
AU  - Yoko Fujita
AU  - Masato Sasaki
AU  - Akiko Kasahara
AU  - Isao Yasumatsu
AU  - Makoto Hirasawa
AU  - Wataru Saitoh
PY  - 2026
JO  - ACS Medicinal Chemistry
Letters
DO  - 10.1021/acsmedchemlett.6c00366
UR  - https://doi.org/10.1021/acsmedchemlett.6c00366
ER  - 

APA

Ogawa, Y., Saito, K., Nakajima, K., Iwamoto, O., Aoki, K., Makino, M., Tanaka, S., Kurikawa, N., Michishita-Kioi, E., Nagata, S., Fujita, Y., Sasaki, M., Kasahara, A., Yasumatsu, I., Hirasawa, M., & Saitoh, W. (2026). Discovery of Forvisirvat (DS-7830a/SP-624), a Brain-Penetrant Sirtuin 6 Activator Derived from Griseofulvin with Antidepressant-Like Effects. ACS Medicinal Chemistry Letters. https://doi.org/10.1021/acsmedchemlett.6c00366

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