Identification, Structure-Activity Relationship (SAR), and Biological Evaluation of New Chemical Series as Malaria Parasite PfGCN5 Bromodomain Inhibitors.

Martin-Acosta P, Al Temimi AHK, Godoy Magalhaes L, Salamanca-Viloria J, Martin Hernando JI, Villegas AI, Franco Hidalgo V, McMillan J, Plater A, Anderson M, Gabarro R, Calderon F, Martinez-Martinez MS, D'Oria E, Siqueira-Neto JL, Forte B, Fernandez E, Winzeler EA, Valenciano AL, Baragaña B, Moliner-Cubel S, Gamo FJ

Open source

DOI: 10.1021/acsomega.6c08259
Published: 2026 Sep 15
Container: ACS omega
Publisher: Not recorded
Open access: yes

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Cite this work

BibTeX

@article{allodium:10.1021/acsomega.6c08259,
  title = {Identification, Structure-Activity Relationship (SAR), and Biological Evaluation of New Chemical Series as Malaria Parasite PfGCN5 Bromodomain Inhibitors.},
  author = {Martin-Acosta P and Al Temimi AHK and Godoy Magalhaes L and Salamanca-Viloria J and Martin Hernando JI and Villegas AI and Franco Hidalgo V and McMillan J and Plater A and Anderson M and Gabarro R and Calderon F and Martinez-Martinez MS and D'Oria E and Siqueira-Neto JL and Forte B and Fernandez E and Winzeler EA and Valenciano AL and Baragaña B and Moliner-Cubel S and Gamo FJ},
  year = {2026},
  journal = {ACS omega},
  doi = {10.1021/acsomega.6c08259},
  url = {https://doi.org/10.1021/acsomega.6c08259}
}

RIS

TY  - JOUR
TI  - Identification, Structure-Activity Relationship (SAR), and Biological Evaluation of New Chemical Series as Malaria Parasite PfGCN5 Bromodomain Inhibitors.
AU  - Martin-Acosta P
AU  - Al Temimi AHK
AU  - Godoy Magalhaes L
AU  - Salamanca-Viloria J
AU  - Martin Hernando JI
AU  - Villegas AI
AU  - Franco Hidalgo V
AU  - McMillan J
AU  - Plater A
AU  - Anderson M
AU  - Gabarro R
AU  - Calderon F
AU  - Martinez-Martinez MS
AU  - D'Oria E
AU  - Siqueira-Neto JL
AU  - Forte B
AU  - Fernandez E
AU  - Winzeler EA
AU  - Valenciano AL
AU  - Baragaña B
AU  - Moliner-Cubel S
AU  - Gamo FJ
PY  - 2026
JO  - ACS omega
DO  - 10.1021/acsomega.6c08259
UR  - https://doi.org/10.1021/acsomega.6c08259
ER  -

APA

P, M., AHK, A. T., L, G. M., J, S., JI, M. H., AI, V., V, F. H., J, M., A, P., M, A., R, G., F, C., MS, M., E, D., JL, S., B, F., E, F., EA, W., AL, V., B, B., S, M., & FJ, G. (2026). Identification, Structure-Activity Relationship (SAR), and Biological Evaluation of New Chemical Series as Malaria Parasite PfGCN5 Bromodomain Inhibitors.. ACS omega. https://doi.org/10.1021/acsomega.6c08259

Source records

pubmed · retrieved 2026-09-25T08:53:26.223Z