β-d-Arabinofuranose-configured Cyclitol Aziridines as Selective, Brain-penetrant Covalent GBA2 Inhibitors.

Lammers RF, Su Q, Mazo L, A Offen W, Ottenhoff R, Bulterman MJ, van der Lienden M, Ferraz MJ, Küllmer F, Ilhan Z, van den Elst H, van der Made I, van Roomen CPAA, de Jongh A, van den Nieuwendijk AMCH, Boot RG, Zelcer N, Davies GJ, Rovira C, Overkleeft HS, Aerts JMFG, Artola M

Open source

DOI
10.1021/jacs.6c09754
Published
2026 Oct 14
Container
Journal of the American Chemical Society
Publisher
Not recorded
Open access
yes

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BibTeX

@article{allodium:10.1021/jacs.6c09754,
  title = {β-d-Arabinofuranose-configured Cyclitol Aziridines as Selective, Brain-penetrant Covalent GBA2 Inhibitors.},
  author = {Lammers RF and Su Q and Mazo L and A Offen W and Ottenhoff R and Bulterman MJ and van der Lienden M and Ferraz MJ and Küllmer F and Ilhan Z and van den Elst H and van der Made I and van Roomen CPAA and de Jongh A and van den Nieuwendijk AMCH and Boot RG and Zelcer N and Davies GJ and Rovira C and Overkleeft HS and Aerts JMFG and Artola M},
  year = {2026},
  journal = {Journal of the American Chemical Society},
  doi = {10.1021/jacs.6c09754},
  url = {https://doi.org/10.1021/jacs.6c09754}
}

RIS

TY  - JOUR
TI  - β-d-Arabinofuranose-configured Cyclitol Aziridines as Selective, Brain-penetrant Covalent GBA2 Inhibitors.
AU  - Lammers RF
AU  - Su Q
AU  - Mazo L
AU  - A Offen W
AU  - Ottenhoff R
AU  - Bulterman MJ
AU  - van der Lienden M
AU  - Ferraz MJ
AU  - Küllmer F
AU  - Ilhan Z
AU  - van den Elst H
AU  - van der Made I
AU  - van Roomen CPAA
AU  - de Jongh A
AU  - van den Nieuwendijk AMCH
AU  - Boot RG
AU  - Zelcer N
AU  - Davies GJ
AU  - Rovira C
AU  - Overkleeft HS
AU  - Aerts JMFG
AU  - Artola M
PY  - 2026
JO  - Journal of the American Chemical Society
DO  - 10.1021/jacs.6c09754
UR  - https://doi.org/10.1021/jacs.6c09754
ER  - 

APA

RF, L., Q, S., L, M., W, A. O., R, O., MJ, B., M, V. D. L., MJ, F., F, K., Z, I., H, V. D. E., I, V. D. M., CPAA, V. R., A, D. J., AMCH, V. D. N., RG, B., N, Z., GJ, D., C, R., HS, O., JMFG, A., & M, A. (2026). β-d-Arabinofuranose-configured Cyclitol Aziridines as Selective, Brain-penetrant Covalent GBA2 Inhibitors.. Journal of the American Chemical Society. https://doi.org/10.1021/jacs.6c09754

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