Design and synthesis of [2-(8,9-dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl)-ethyl]phosphonic acid (EAA-090), a potent N-methyl-D-aspartate antagonist, via the use of 3-cyclobutene-1,2-dione as an achiral alpha-amino acid bioisostere.
- DOI
- 10.1021/jm970504g
- Published
- 1998 Jan 15
- Container
- Journal of medicinal chemistry
- Publisher
- Not recorded
- Open access
- unknown
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Cite this work
BibTeX
@article{allodium:10.1021/jm970504g,
title = {Design and synthesis of [2-(8,9-dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl)-ethyl]phosphonic acid (EAA-090), a potent N-methyl-D-aspartate antagonist, via the use of 3-cyclobutene-1,2-dione as an achiral alpha-amino acid bioisostere.},
author = {Kinney WA and Abou-Gharbia M and Garrison DT and Schmid J and Kowal DM and Bramlett DR and Miller TL and Tasse RP and Zaleska MM and Moyer JA},
year = {1998},
journal = {Journal of medicinal chemistry},
doi = {10.1021/jm970504g},
url = {https://doi.org/10.1021/jm970504g}
}RIS
TY - JOUR TI - Design and synthesis of [2-(8,9-dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl)-ethyl]phosphonic acid (EAA-090), a potent N-methyl-D-aspartate antagonist, via the use of 3-cyclobutene-1,2-dione as an achiral alpha-amino acid bioisostere. AU - Kinney WA AU - Abou-Gharbia M AU - Garrison DT AU - Schmid J AU - Kowal DM AU - Bramlett DR AU - Miller TL AU - Tasse RP AU - Zaleska MM AU - Moyer JA PY - 1998 JO - Journal of medicinal chemistry DO - 10.1021/jm970504g UR - https://doi.org/10.1021/jm970504g ER -
APA
WA, K., M, A., DT, G., J, S., DM, K., DR, B., TL, M., RP, T., MM, Z., & JA, M. (1998). Design and synthesis of [2-(8,9-dioxo-2,6-diazabicyclo[5.2.0]non-1(7)-en-2-yl)-ethyl]phosphonic acid (EAA-090), a potent N-methyl-D-aspartate antagonist, via the use of 3-cyclobutene-1,2-dione as an achiral alpha-amino acid bioisostere.. Journal of medicinal chemistry. https://doi.org/10.1021/jm970504g
Source records
- pubmed · retrieved 2026-09-25T13:13:44.025Z