Potent and selective bivalent inhibitors of BET bromodomains.

Waring MJ, Chen H, Rabow AA, Walker G, Bobby R, Boiko S, Bradbury RH, Callis R, Clark E, Dale I, Daniels DL, Dulak A, Flavell L, Holdgate G, Jowitt TA, Kikhney A, McAlister M, Méndez J, Ogg D, Patel J, Petteruti P, Robb GR, Robers MB, Saif S, Stratton N, Svergun DI, Wang W, Whittaker D, Wilson DM, Yao Y

Open source

DOI: 10.1038/nchembio.2210
Published: 2016 Dec
Container: Nature chemical biology
Publisher: Not recorded
Open access: unknown

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Cite this work

BibTeX

@article{allodium:10.1038/nchembio.2210,
  title = {Potent and selective bivalent inhibitors of BET bromodomains.},
  author = {Waring MJ and Chen H and Rabow AA and Walker G and Bobby R and Boiko S and Bradbury RH and Callis R and Clark E and Dale I and Daniels DL and Dulak A and Flavell L and Holdgate G and Jowitt TA and Kikhney A and McAlister M and Méndez J and Ogg D and Patel J and Petteruti P and Robb GR and Robers MB and Saif S and Stratton N and Svergun DI and Wang W and Whittaker D and Wilson DM and Yao Y},
  year = {2016},
  journal = {Nature chemical biology},
  doi = {10.1038/nchembio.2210},
  url = {https://doi.org/10.1038/nchembio.2210}
}

RIS

TY  - JOUR
TI  - Potent and selective bivalent inhibitors of BET bromodomains.
AU  - Waring MJ
AU  - Chen H
AU  - Rabow AA
AU  - Walker G
AU  - Bobby R
AU  - Boiko S
AU  - Bradbury RH
AU  - Callis R
AU  - Clark E
AU  - Dale I
AU  - Daniels DL
AU  - Dulak A
AU  - Flavell L
AU  - Holdgate G
AU  - Jowitt TA
AU  - Kikhney A
AU  - McAlister M
AU  - Méndez J
AU  - Ogg D
AU  - Patel J
AU  - Petteruti P
AU  - Robb GR
AU  - Robers MB
AU  - Saif S
AU  - Stratton N
AU  - Svergun DI
AU  - Wang W
AU  - Whittaker D
AU  - Wilson DM
AU  - Yao Y
PY  - 2016
JO  - Nature chemical biology
DO  - 10.1038/nchembio.2210
UR  - https://doi.org/10.1038/nchembio.2210
ER  -

APA

MJ, W., H, C., AA, R., G, W., R, B., S, B., RH, B., R, C., E, C., I, D., DL, D., A, D., L, F., G, H., TA, J., A, K., M, M., J, M., D, O., J, P., P, P., GR, R., MB, R., S, S., N, S., DI, S., W, W., D, W., DM, W., & Y, Y. (2016). Potent and selective bivalent inhibitors of BET bromodomains.. Nature chemical biology. https://doi.org/10.1038/nchembio.2210

Source records

pubmed · retrieved 2026-09-25T19:19:16.501Z