Selective inhibitors of SARM1 targeting an allosteric cysteine in the autoregulatory ARM domain

Hannah C. Feldman, Elisa Merlini, Carlos Guijas, Kristen E. DeMeester, Evert Njomen, Ellen M. Kozina, Minoru Yokoyama, Ekaterina Vinogradova, Holly T. Reardon, Bruno Melillo, Stuart L. Schreiber, Andrea Loreto, Jacqueline L. Blankman, Benjamin F. Cravatt

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DOI
10.1073/pnas.2208457119
Published
2022-08-22
Container
Proceedings of the National Academy of Sciences
Publisher
National Academy of Sciences
Open access
unknown

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BibTeX

@article{allodium:10.1073/pnas.2208457119,
  title = {Selective inhibitors of SARM1 targeting an allosteric cysteine in the autoregulatory ARM domain},
  author = {Hannah C. Feldman and Elisa Merlini and Carlos Guijas and Kristen E. DeMeester and Evert Njomen and Ellen M. Kozina and Minoru Yokoyama and Ekaterina Vinogradova and Holly T. Reardon and Bruno Melillo and Stuart L. Schreiber and Andrea Loreto and Jacqueline L. Blankman and Benjamin F. Cravatt},
  year = {2022},
  journal = {Proceedings of the National Academy of Sciences},
  doi = {10.1073/pnas.2208457119},
  url = {https://doi.org/10.1073/pnas.2208457119}
}

RIS

TY  - JOUR
TI  - Selective inhibitors of SARM1 targeting an allosteric cysteine in the autoregulatory ARM domain
AU  - Hannah C. Feldman
AU  - Elisa Merlini
AU  - Carlos Guijas
AU  - Kristen E. DeMeester
AU  - Evert Njomen
AU  - Ellen M. Kozina
AU  - Minoru Yokoyama
AU  - Ekaterina Vinogradova
AU  - Holly T. Reardon
AU  - Bruno Melillo
AU  - Stuart L. Schreiber
AU  - Andrea Loreto
AU  - Jacqueline L. Blankman
AU  - Benjamin F. Cravatt
PY  - 2022
JO  - Proceedings of the National Academy of Sciences
DO  - 10.1073/pnas.2208457119
UR  - https://doi.org/10.1073/pnas.2208457119
ER  - 

APA

Feldman, H. C., Merlini, E., Guijas, C., DeMeester, K. E., Njomen, E., Kozina, E. M., Yokoyama, M., Vinogradova, E., Reardon, H. T., Melillo, B., Schreiber, S. L., Loreto, A., Blankman, J. L., & Cravatt, B. F. (2022). Selective inhibitors of SARM1 targeting an allosteric cysteine in the autoregulatory ARM domain. Proceedings of the National Academy of Sciences. https://doi.org/10.1073/pnas.2208457119

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