Dasatinib (BMS-354825), a dual SRC/ABL kinase inhibitor, inhibits the kinase activity of wild-type, juxtamembrane, and activation loop mutant KIT isoforms associated with human malignancies.

Schittenhelm MM, Shiraga S, Schroeder A, Corbin AS, Griffith D, Lee FY, Bokemeyer C, Deininger MW, Druker BJ, Heinrich MC

Open source

DOI
10.1158/0008-5472.can-05-2050
Published
2006 Jan 1
Container
Cancer research
Publisher
Not recorded
Open access
unknown

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BibTeX

@article{allodium:10.1158/0008-5472.can-05-2050,
  title = {Dasatinib (BMS-354825), a dual SRC/ABL kinase inhibitor, inhibits the kinase activity of wild-type, juxtamembrane, and activation loop mutant KIT isoforms associated with human malignancies.},
  author = {Schittenhelm MM and Shiraga S and Schroeder A and Corbin AS and Griffith D and Lee FY and Bokemeyer C and Deininger MW and Druker BJ and Heinrich MC},
  year = {2006},
  journal = {Cancer research},
  doi = {10.1158/0008-5472.can-05-2050},
  url = {https://doi.org/10.1158/0008-5472.can-05-2050}
}

RIS

TY  - JOUR
TI  - Dasatinib (BMS-354825), a dual SRC/ABL kinase inhibitor, inhibits the kinase activity of wild-type, juxtamembrane, and activation loop mutant KIT isoforms associated with human malignancies.
AU  - Schittenhelm MM
AU  - Shiraga S
AU  - Schroeder A
AU  - Corbin AS
AU  - Griffith D
AU  - Lee FY
AU  - Bokemeyer C
AU  - Deininger MW
AU  - Druker BJ
AU  - Heinrich MC
PY  - 2006
JO  - Cancer research
DO  - 10.1158/0008-5472.can-05-2050
UR  - https://doi.org/10.1158/0008-5472.can-05-2050
ER  - 

APA

MM, S., S, S., A, S., AS, C., D, G., FY, L., C, B., MW, D., BJ, D., & MC, H. (2006). Dasatinib (BMS-354825), a dual SRC/ABL kinase inhibitor, inhibits the kinase activity of wild-type, juxtamembrane, and activation loop mutant KIT isoforms associated with human malignancies.. Cancer research. https://doi.org/10.1158/0008-5472.can-05-2050

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