Potent and selective bivalent inhibitors of BET bromodomains

Michael Waring, H Chen, AA Rabow, G Walker, R Bobby, S Boiko, RH Bradbury, R Callis, E Clark, E Dale, DL Daniels, A Dulak, L Flavell, G Holdgate, TA Jowitt, A Kikhney, M McAlister, J Mendez, D Ogg, J Patel, P Petteruti, GR Robb, MB Robers, S Saif, N Stratton, DI Svergun, W Wang, D Whittaker, DM Wilson, Y Yao

Open source

DOI: 10.25405/ncl.34280541.v1
Published: 2026
Container: Not recorded
Publisher: Newcastle University
Open access: yes

Credibility signals

limited evidence Score 47/100 under policy 1.0.0. This is a metadata assessment, not a judgment of the paper's conclusions.

Show all credibility signals

cautionDOI registered: No matching Crossref record was present in this response. Source: Crossref; license: CC0 metadata
cautionDOI resolves: No matching Crossref record was present in this response. Source: Crossref; license: CC0 metadata
not scoredDirectory of Open Access Journals: No matching DOAJ record was present in this response. No allow-list match; this is not evidence of low credibility. Source: DOAJ; license: CC0
not scoredMEDLINE indexed: Not checked or no result supplied; no credibility inference made. Source: No authority result supplied; license: Unknown
not scoredOpenAlex core source: Not checked or no result supplied; no credibility inference made. Source: No authority result supplied; license: Unknown
not scoredKnown publisher allow-list: Not checked or no result supplied; no credibility inference made. Source: No authority result supplied; license: Unknown
not scoredROR affiliation: Not checked or no result supplied; no credibility inference made. Source: No authority result supplied; license: Unknown
not scoredRetraction Watch retraction: No retraction notice matched this DOI in the deployed snapshot. No matching event found; coverage may be incomplete. Source: Retraction Watch; license: CC BY 4.0
not scoredRetraction Watch expression of concern: No expression of concern notice matched this DOI in the deployed snapshot. No matching event found; coverage may be incomplete. Source: Retraction Watch; license: CC BY 4.0
not scoredRetraction Watch correction: No correction notice matched this DOI in the deployed snapshot. No matching event found; coverage may be incomplete. Source: Retraction Watch; license: CC BY 4.0
not scoredRetraction Watch reinstatement: No reinstatement notice matched this DOI in the deployed snapshot. No matching event found; coverage may be incomplete. Source: Retraction Watch; license: CC BY 4.0
supportingOpen access status: Normalized open-access status: open. Source: Normalized work metadata; license: Caller-provided; provenance license not supplied to scorer
supportingPublication license: A publication license was supplied: https://creativecommons.org/licenses/by-nc/4.0/legalcode. Presence improves reuse transparency, not research validity. Source: Normalized work metadata; license: Caller-provided; provenance license not supplied to scorer
not scoredPublication version: A publication version was supplied but is not scored. Source: Normalized work metadata; license: Caller-provided; provenance license not supplied to scorer
cautionMetadata completeness: 5 of 6 scored descriptive metadata groups are present; missing fields increase uncertainty. Source: Normalized work metadata; license: Caller-provided; provenance license not supplied to scorer

Cite this work

BibTeX

@article{allodium:10.25405/ncl.34280541.v1,
  title = {Potent and selective bivalent inhibitors of BET bromodomains},
  author = {Michael Waring and H Chen and AA Rabow and G Walker and R Bobby and S Boiko and RH Bradbury and R Callis and E Clark and E Dale and DL Daniels and A Dulak and L Flavell and G Holdgate and TA Jowitt and A Kikhney and M McAlister and J Mendez and D Ogg and J Patel and P Petteruti and GR Robb and MB Robers and S Saif and N Stratton and DI Svergun and W Wang and D Whittaker and DM Wilson and Y Yao},
  year = {2026},
  doi = {10.25405/ncl.34280541.v1},
  url = {https://doi.org/10.25405/ncl.34280541.v1}
}

RIS

TY  - JOUR
TI  - Potent and selective bivalent inhibitors of BET bromodomains
AU  - Michael Waring
AU  - H Chen
AU  - AA Rabow
AU  - G Walker
AU  - R Bobby
AU  - S Boiko
AU  - RH Bradbury
AU  - R Callis
AU  - E Clark
AU  - E Dale
AU  - DL Daniels
AU  - A Dulak
AU  - L Flavell
AU  - G Holdgate
AU  - TA Jowitt
AU  - A Kikhney
AU  - M McAlister
AU  - J Mendez
AU  - D Ogg
AU  - J Patel
AU  - P Petteruti
AU  - GR Robb
AU  - MB Robers
AU  - S Saif
AU  - N Stratton
AU  - DI Svergun
AU  - W Wang
AU  - D Whittaker
AU  - DM Wilson
AU  - Y Yao
PY  - 2026
DO  - 10.25405/ncl.34280541.v1
UR  - https://doi.org/10.25405/ncl.34280541.v1
ER  -

APA

Waring, M., Chen, H., Rabow, A., Walker, G., Bobby, R., Boiko, S., Bradbury, R., Callis, R., Clark, E., Dale, E., Daniels, D., Dulak, A., Flavell, L., Holdgate, G., Jowitt, T., Kikhney, A., McAlister, M., Mendez, J., Ogg, D., Patel, J., Petteruti, P., Robb, G., Robers, M., Saif, S., Stratton, N., Svergun, D., Wang, W., Whittaker, D., Wilson, D., & Yao, Y. (2026). Potent and selective bivalent inhibitors of BET bromodomains. https://doi.org/10.25405/ncl.34280541.v1

Source records

datacite · retrieved 2026-11-10T13:27:30.093Z