AS-LRRK2 & AS-SYN Series Version 2.8.0: Multi-Vector Parkinson's Disease Platform (2026) — De Novo LRRK2 G2019S Kinase Inhibitors (AS-LRRK2-006B-DualD4, AS-LRRK2-Pyr-Spiro-v2, AS-LRRK2-006A-DualD4), First-in-Class Alpha-Synuclein Oligomerization Inhibitors (AS-SYN-003 & AS-SYN-007-TriOCD3), Two-Layer Selectivity Paradigm (240x-431x in silico vs 20x-50x cellular), and Independent SIB SwissADME Audit

Sokolov, Artyom

Open source

DOI
10.5281/zenodo.23526889
Published
2026
Container
Not recorded
Publisher
Zenodo
Open access
yes

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BibTeX

@article{allodium:10.5281/zenodo.23526889,
  title = {AS-LRRK2 \& AS-SYN Series Version 2.8.0: Multi-Vector Parkinson's Disease Platform (2026) — De Novo LRRK2 G2019S Kinase Inhibitors (AS-LRRK2-006B-DualD4, AS-LRRK2-Pyr-Spiro-v2, AS-LRRK2-006A-DualD4), First-in-Class Alpha-Synuclein Oligomerization Inhibitors (AS-SYN-003 \& AS-SYN-007-TriOCD3), Two-Layer Selectivity Paradigm (240x-431x in silico vs 20x-50x cellular), and Independent SIB SwissADME Audit},
  author = {Sokolov, Artyom},
  year = {2026},
  doi = {10.5281/zenodo.23526889},
  url = {https://doi.org/10.5281/zenodo.23526889}
}

RIS

TY  - JOUR
TI  - AS-LRRK2 & AS-SYN Series Version 2.8.0: Multi-Vector Parkinson's Disease Platform (2026) — De Novo LRRK2 G2019S Kinase Inhibitors (AS-LRRK2-006B-DualD4, AS-LRRK2-Pyr-Spiro-v2, AS-LRRK2-006A-DualD4), First-in-Class Alpha-Synuclein Oligomerization Inhibitors (AS-SYN-003 & AS-SYN-007-TriOCD3), Two-Layer Selectivity Paradigm (240x-431x in silico vs 20x-50x cellular), and Independent SIB SwissADME Audit
AU  - Sokolov, Artyom
PY  - 2026
DO  - 10.5281/zenodo.23526889
UR  - https://doi.org/10.5281/zenodo.23526889
ER  - 

APA

Artyom, S. (2026). AS-LRRK2 & AS-SYN Series Version 2.8.0: Multi-Vector Parkinson's Disease Platform (2026) — De Novo LRRK2 G2019S Kinase Inhibitors (AS-LRRK2-006B-DualD4, AS-LRRK2-Pyr-Spiro-v2, AS-LRRK2-006A-DualD4), First-in-Class Alpha-Synuclein Oligomerization Inhibitors (AS-SYN-003 & AS-SYN-007-TriOCD3), Two-Layer Selectivity Paradigm (240x-431x in silico vs 20x-50x cellular), and Independent SIB SwissADME Audit. https://doi.org/10.5281/zenodo.23526889

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